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Faculty members

Content

Inside a building, a man dressed in a traditional white uniform with a red and white Saudi shemagh wears a neutral expression as if he were taking a picture of a faculty file at Qassim University.
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KAIS IBRAHIM MOHAMED AOUADI

Full Professor
College of Sciences
Chemistry Department

Personal data

  • K.AOUADI@qu.edu.sa
  • Desktop watches
    Google Scholar
    OneDrive

    Scientific qualifications

    • University Qualification Certificate (UQC)
    • PhD specializing in organic chemistry
    • Master of Organic Chemistry
    • Professorship

    Research interests

    • Amino Acid Synthesis
    • 3,1-bipolar cyclic addition
    • Synthesis of chiral isoxazolidinediones
    • Heterogeneous ring manufacturing
    • https://scholar.google.com/citations?user=x9N7hO4AAAAJ&hl=fr

    Published research

    • An untargeted metabolomics approach based on UPLC-ESI-QTOF-MS/MS and an evaluation of the antioxidant and cytotoxic activities of Nepeta deflersiana Schweinf. ex Hedge, supported by molecular modeling and ADMET analysis (2025-01-18)
    • Exploring the antioxidant potency of novel indolin-2-one-based imidazo-isoxazole hybrids: Design, synthesis, and computational studies (2025-10-02)
    • Anti-ulcer Activity of Synthetically Produced Green Selenium Nanoparticles Using Nigella sativa L. Seed Extract in Rats (2025-11-21)
    • Synthesis, Structure-Activity Relationship and in silico Studies of Novel Pyrazolothiazole and Thiazolopyridine Derivatives as Prospective Antimicrobial and Anticancer Agents (2021-08-20)
    • Bioactivities and in silico study of the phytochemicals of Pergularia tomentosa L. as potent antimicrobial agents targeting type IIA topoisomerase, TyrRS, and Sap1 virulence proteins (2021-01-17)
    • Design, Synthesis, ADMET, and Molecular Docking of New Imidazo[4,5-b]pyridine-5-thione Derivatives as Potential Tyrosyl-tRNA Synthetase Inhibitors (2020-09-01)
    • New substituted pyrazolones and dipyrazolotriazines as promising tyrosyl-tRNA synthetase and peroxiredoxin-5 inhibitors: Design, synthesis, molecular docking, and structure-activity relationship (SAR) analysis (2021-02-17)
    • Novel fused pyridine derivatives containing a pyrimidine moiety as prospective tyrosyl-tRNA synthetase inhibitors: Design, synthesis, pharmacokinetics, and molecular docking studies (2020-11-05)
    • Toward a Treatment for Antibacterial and Antifungal Infections: Design, Synthesis, and In Vitro Activity of Novel Arylhydrazothiazolylsulfonamide Analogs and Insights from DFT, Docking, and Molecular Dynamics Simulations (2021-06-20)
    • New Spiropyrrolothiazole Derivatives Bearing an Oxazolone Moiety as Potential Antidiabetic Agents: Design, Synthesis, Crystal Structure, Hirshfeld Surface Analysis, ADME, and Molecular Docking Studies (2022-01-17)
    • Novel (2-Oxoindolin-3-ylidene)methyl)-1H-pyrazole and Their Fused Derivatives: Design, Synthesis, Antimicrobial Evaluation, DFT, Chemical Approach, In Silico ADME, and Molecular Docking Studies (2022-05-24)
    • Design, synthesis, in vitro anticancer and antimicrobial evaluation, SAR analysis, molecular docking, and dynamic simulation of new isoxazole derivatives based on pyrazoles, triazoles, and pyridazines (2022-05-23)
    • Effect of the coordination of the π-acceptor 4-cyanopyridine ligand on the structural and electronic properties of meso-tetra(para-methoxy) and meso-tetra(para-chlorophenyl) porphyrin cobalt(II) coordination compounds. Application in the catalytic degradation of methylene blue dye (2020-02-17)
    • Zinc(II) triazole-meso-aryl-substituted porphyrins for UV-visible detection of chloride and bromide. Adsorption and catalytic degradation of malachite green dye (2020-06-14)
    • Emetine, A Potent Alkaloid for the Treatment of SARS-CoV-2 Targeting Papain-like Protease and Non-structural Proteins: Pharmacokinetics, Molecular Docking, and Dynamic Studies (2022-01-01)
    • Phytochemical profiling, antimicrobial, antibiofilm, insecticidal, and anti-leishmanial properties of an aqueous extract from the root bark of Juglans regia L.: In vitro and in silico approaches (2023-12-31)
    • Tripeptides from Allium subhirsitum L. extracts: Pharmacokinetic properties, toxicity prediction, and in silico study against SARS-CoV-2 enzymes and pro-inflammatory proteins (2021-01-01)
    • Repurposing of anisomycin and oleandomycin as potential anti-SARS-CoV-2 virus agents targeting key enzymes using virtual computational approaches (2021-01-01)
    • Preparation and characterization of ZnO nanoparticles incorporated by mechanical milling into cellulose for electrical insulator applications (2022-04-01)
    • GC-MS/MS Analysis and Wound-Healing Potential of Urtica dioica Essential Oil: In Silico Modeling and an In Vivo Study in Rats (2024-07-05)
    • LC-ESI/MS Phytochemical Profiling and the Antioxidant, Antibacterial, Antifungal, Antiviral, and In Silico Pharmacological Properties of Organic Extracts from Algerian Asphodelus tenuifolius (Cav.) (2021-04-01)
    • Allium subhirsutum L. as a Potential Source of Antioxidant and Anticancer Bioactive Molecules: HR-LCMS Phytochemical Profiling, In Vitro and In Vivo Pharmacological Study (2020-10-01)
    • HR-LCMS-Based Metabolite Profiling, Antioxidant, and Anticancer Properties of the Methanolic Extract of Teucrium polium L.: A Computational and In Vitro Study (2020-11-01)
    • Tomatidine and Patchouli Alcohol as Inhibitors of SARS-CoV-2 Enzymes (3CLpro, PLpro, and NSP15) by Molecular Docking and Molecular Dynamics Simulations (2021-10-01)
    • Antimicrobial, Antioxidant, Anti-Acetylcholinesterase, Antidiabetic, and Pharmacokinetic Properties of Carum carvi L. and Coriandrum sativum L. Essential Oils, Alone and in Combination (2021-06-01)
    • Lapachol and (α/β)-Lapachone as Inhibitors of SARS-CoV-2 Main Protease (Mpro) and hACE-2: ADME Properties, Docking, and Dynamic Simulation Approaches (2022-07-01)
    • Optical and photoelectronic properties of a new material: Optoelectronic application (2020-01-01)
    • Antioxidant Activities of a New Chemotype of Piper cubeba L. Fruit Essential Oil (Methyleugenol/Eugenol): In Silico Molecular Docking and ADMET Studies (2020-11-01)
    • Antimicrobial, Antioxidant, Anti-Acetylcholinesterase, Antidiabetic, and Pharmacokinetic Properties of Carum carvi L. and Coriandrum sativum L. Essential Oils … (2021-01-01)
    • Antioxidant Activities of a New Chemotype of *Piper cubeba* L. Fruit Essential Oil (Methyleugenol/Eugenol): In Silico Molecular Docking and ADMET Studies (2020-01-01)
    • Tomatidine and patchouli alcohol as inhibitors of SARS-CoV-2 enzymes (3CLpro, PLpro, and NSP15) by molecular docking and molecular dynamics simulations (2021-01-01)
    • Toward a treatment of antibacterial and antifungal infections: Design, synthesis, and in vitro activity of novel arylhydrazothiazolylsulfonamide analogues and their insight into… (2021-01-01)
    • Synthesis, in vitro antimicrobial assessment, and computational investigation of pharmacokinetic and bioactivity properties of novel trifluoromethylated compounds using in … (2020-01-01)
    • In vitro antimicrobial and α-glucosidase inhibitory potential of enantiopure cycloalkylglycine derivatives: Insights into their in silico pharmacokinetic, druglikeness, and … (2020-01-01)
    • HR-LCMS-Based Metabolite Profiling, Antioxidant, and Anticancer Properties of Teucrium polium L. Methanolic Extract: Computational and In Vitro Study (2020-01-01)
    • Divergent synthesis of a pochonin library targeting HSP90 and in vivo efficacy of identified inhibitor (2008-01-01)
    • Design, synthesis, in vitro anticancer and antimicrobial evaluation, SAR analysis, molecular docking and dynamic simulation of new pyrazoles, triazoles, and pyridazines based … (2022-01-01)
    • Allium subhirsutum L. as a Potential Source of Antioxidant and Anticancer Bioactive Molecules: HR-LCMS Phytochemical Profiling, In Vitro and In Vivo … (2020-01-01)
    • Design, synthesis, molecular properties, and in vitro antioxidant and antibacterial potential of novel enantiopure isoxazolidine derivatives (2020-01-01)
    • Novel fused pyridine derivatives containing a pyrimidine moiety as prospective tyrosyl-tRNA synthetase inhibitors: Design, synthesis, pharmacokinetics, and molecular docking studies (2020-01-01)
    • Synthesis, structure-activity relationship, and in silico studies of novel pyrazolothiazole and thiazolopyridine derivatives as prospective antimicrobial and anticancer agents (2021-01-01)
    • Inhibition of HSP90 with Pochoximes: SAR and Structure-Based Insights (2009-01-01)
    • Design, synthesis, biological evaluation, and in silico studies of novel 1, 2, 3-triazole-linked benzoxazine-2,4-dione conjugates as potent antimicrobial, antioxidant, and anti… (2022-01-01)
    • Stereoselective synthesis of enantiopure N-substituted pyrrolidine-2,5-dione derivatives via 1,3-dipolar cycloaddition and assessment of their in vitro antioxidant and ... (2017-01-01)
    • Multifunctional isoxazolidine derivatives as α-amylase and α-glucosidase inhibitors (2020-01-01)
    • Design, synthesis, ADMET, and molecular docking of new imidazo[4,5-b]pyridine-5-thione derivatives as potential tyrosyl-tRNA synthetase inhibitors (2020-01-01)
    • Effect of the coordination of $\pi$-acceptor 4-cyanopyridine ligand on the structural and electronic properties of meso-tetra($p$-methoxyphenyl) and meso-tetra($p$-chlorophenyl porphyrins (2020-01-01)
    • GC/MS Profiling, Antibacterial, Anti-Quorum Sensing, and Antibiofilm Properties of Anethum graveolens L. Essential Oil: Molecular Docking Study and In-Silico ... (2023-01-01)
    • GC-MS Profiling, Vibriocidal, Antioxidant, Antibiofilm, and Anti-Quorum Sensing Properties of Carum carvi L. Essential Oil: In Vitro and In Silico Approaches (2022-01-01)
    • 1,3-Dipolar cycloaddition of a chiral nitrone to (E)-1,4-dichloro-2-butene: a new efficient synthesis of (2S,3S,4R)-4-hydroxyisoleucine (2012-01-01)
    • New substituted pyrazolones and dipyrazolotriazines as promising tyrosyl-tRNA synthetase and peroxiredoxin-5 inhibitors: Design, synthesis, molecular docking, and structure… (2021-01-01)
    • Novel enantiopure isoxazolidine and C-alkyl imine oxide derivatives as potential hypoglycemic agents: Design, synthesis, dual inhibitors of α-amylase and α-glucosidase, ADMET ... (2020-01-01)
    • Analogues of insulin secretagogue (2S, 3R, 4S)-4-hydroxyisoleucine: synthesis by 1,3-dipolar cycloaddition reactions of chiral nitrones to alkenes (2008-01-01)
    • HPLC/MS Phytochemical Profiling with Antioxidant Activities of Echium humile Desf. Extracts: ADMET Prediction and Computational Study Targeting Human … (2021-01-01)
    • Unprecedented stereoselective synthesis of 3-methylisoxazolidin-5-aryl-1,2,4-oxadiazoles via 1,3-dipolar cycloaddition and study of their in vitro antioxidant activity (2016-01-01)
    • Cycloadditions of chiral nitrones to racemic 3-substituted butenes: a direct access with kinetic resolution to enantiopure dihydroxylated amino acids (2006-01-01)
    • Multifunctional derivatives of spiropyrrolidine tethered indeno-quinoxaline heterocyclic hybrids as potent antimicrobial, antioxidant, and antidiabetic agents: design, synthesis… (2022-01-01)
    • In Vitro and In Silico Screening of Anti-Vibrio spp., Antibiofilm, Antioxidant and Anti-Quorum Sensing Activities of Cuminum cyminum L. Volatile Oil (2022-01-01)
    • LC-ESI/MS-Phytochemical Profiling with Antioxidant, Antibacterial, Antifungal, Antiviral, and In Silico Pharmacological Properties of Algerian Asphodelus Tenuifolius (Cav… (2021-01-01)
    • Cycloaddition of a chiral nitrone to allylic motifs: an access to enantiopure sugar-based amino acids displaying a stable glycosidic bond and to (4S)-4-hydroxy-L-ornithine (2012-01-01)
    • Phytochemical Profiling of *Allium subhirsutum* L. Aqueous Extract with Antioxidant, Antimicrobial, Antibiofilm, and Anti-Quorum Sensing Properties: In Vitro and In … (2022-01-01)
    • Bioactivities and in silico study of Pergularia tomentosa L. phytochemicals as potent antimicrobial agents targeting type IIA topoisomerase, TyrRS, and Sap1 … (2021-01-01)
    • Zinc(II) triazole meso-aryl-substituted porphyrins for UV-visible chloride and bromide detection. Adsorption and catalytic degradation of malachite green dye. (2020-01-01)
    • New synthetic routes toward enantiopure (2S, 3R, 4R)-4-hydroxyisoleucine by 1,3-dipolar cycloaddition of a chiral nitrone to C4 alkenes (2007-01-01)
    • In vitro and in silico evaluation of antiproliferative activity of new isoxazolidine derivatives targeting EGFR: design, synthesis, cell cycle analysis, and apoptotic inducers (2023-01-01)
    • In silico design, synthesis, and evaluation of novel enantiopure isoxazolidines as promising dual inhibitors of α-amylase and α-glucosidase (2024-01-01)
    • Emetine, a potent alkaloid for the treatment of SARS-CoV-2 targeting papain-like protease and non-structural proteins: pharmacokinetics, molecular docking and dynamic studies (2022-01-01)
    • Design, synthesis, and in vitro evaluation of isoxazolidine-isatin hybrids targeting two pathways for antidiabetic potential, along with multiscale molecular modeling approaches. (2024-01-01)
    • Phytochemical Profiling, Antimicrobial, Antibiofilm, Insecticidal, and Anti-Leishmanial Properties of Aqueous Extract from Juglans regia L. Root Bark: In Vitro and In Silico … (2023-01-01)
    • GC-MS/MS Analysis and Wound Repair Potential of Urtica dioica Essential Oil: In silico Modeling and In vivo Study in Rats (2025-01-01)
    • Synthesis, optical properties, DNA, β-cyclodextrin interaction, hydrogen isotope sensor, and computational study of a new enantiopure isoxazolidine derivative (ISoXD) (2024-01-01)
    • New Spiropyrrolothiazole Derivatives Bearing an Oxazolone Moiety as Potential Antidiabetic Agents: Design, Synthesis, Crystal Structure, Hirshfeld Surface Analysis, ADME, and… (2022-01-01)
    • HPLC-MS Profiling, Antioxidant, Antimicrobial, Antidiabetic, and Cytotoxicity Activities of Arthrocnemum indicum (Willd.) Moq. Extracts (2022-01-01)
    • Biological Activities Evaluation of Enantiopure Isoxazolidine Derivatives: In Vitro, In Vivo, and In Silico Studies (2019-01-01)
    • (2-Oxoindolin-3-ylidene)methyl)-1H-pyrazole and their fused derivatives: Design, synthesis, antimicrobial evaluation, DFT, chemical approach, in silico ADME and … (2022-01-01)
    • Synthesis of New Porphyrin Complexes: Evaluations on Optical, Electrochemical, and Electronic Properties, and Application as an Optical Sensor (2019-01-01)
    • Stereoselective synthesis of 1,2,3-triazolyl-functionalized isoxazolidines, via two consecutive 1,3-dipolar cycloadditions, as precursors of unnatural amino acids (2013-01-01)
    • A reversible optical sensor film for mercury ion discrimination based on an isoxazolidine derivative and exhibiting pH sensing (2022-01-01)
    • Phytochemical Profiling, Antimicrobial and α-Glucosidase Inhibitory Potential of Phenolic-Enriched Extracts of the Aerial Parts from Echium humile Desf.: In Vitro … (2022-01-01)
    • X-ray molecular structure characterization of a hexamethylenetetramine zinc(II) porphyrin complex: Catalytic degradation of toluidine blue dye, experimental and statistical... (2021-01-01)
    • Synthesis and SPAR exploration of new semicarbazone-triazole hybrids in search of potent antioxidant, antibacterial, and antifungal agents (2019-01-01)
    • Design, synthesis, biological evaluation, kinetic studies, and molecular modeling of imidazo-isoxazole derivatives targeting both α-amylase and α-glucosidase inhibitors (2024-01-01)
    • GC-MS profile, α-glucosidase inhibitory potential, antibacterial and antioxidant evaluation of Citrus aurantium (L.) peels essential oil (2021-01-01)
    • Novel routes to either racemic or enantiopure α-amino-(4-hydroxy-pyrrolidin-3-yl) acetic acid derivatives and biological evaluation of a new promising pharmacological scaffold (2015-01-01)
    • Synthesis, optical properties, DNA, β-cyclodextrin interactions, and antioxidant evaluation of a novel isoxazolidine derivative (ISoXD2): A multispectral and computational analysis (2024-01-01)
    • Multi-Step Synthesis and Biological Evaluation of Analogues of Insulin Secretagogue (2S,3R,4S)-4-Hydroxyisoleucine (2009-01-01)
    • Lapachol and (α/β)-lapachone as inhibitors of SARS-CoV-2 Main Protease (Mpro) and hACE-2: ADME properties, docking, and dynamic simulation approaches (2022-01-01)
    • Tripeptides from Allium subhirsutum L. extracts: Pharmacokinetic properties, toxicity prediction, and in silico study against SARS-CoV-2 enzymes and pro-inflammatory proteins (2021-01-01)
    • Unexpected synthesis of aziridines under Cu(I)-catalyzed Kinugasa conditions assisted by microwave irradiation (2016-01-01)
    • Stereoselective Synthesis of Enantiopure Cycloalkylglycines via 1,3-Dipolar Cycloaddition of a Chiral Nitrone to Cycloalkenes (2014-01-01)
    • A Cycloaddition–Cyclization Combined Approach to Enantiopure 3‐Glycinyl‐4‐hydroxypyrrolidines and 3‐Substituted 4‐Hydroxyprolines (2014-01-01)
    • Repurposing of anisomycin and oleandomycin as potential anti-SARS-CoV-2 virus agents targeting key enzymes using virtual computational approaches (2022-01-01)
    • Synthesis of some isoxazolidine and isoxazoline derivatives using nitrone-derived (-)-menthone via 1,3-dipolar cycloaddition with alkenes, alkynes, and cycloalkenes (2016-01-01)
    • Untargeted metabolomics approach based on UPLC-ESI-QTOF-MS/MS and evaluation of antioxidant and cytotoxic activities of Nepeta deflersiana Schweinf. ex Hedge supported by … (2025-01-01)
    • A stereoselective method for the synthesis of enantiopure 3-substituted 4-hydroxyproline derivatives via 1,3-dipolar cycloadditions (2016-01-01)
    • C-glycosyl amino-substituted hydro- and benzoquinones: Synthesis and preliminary biological evaluation (2007-01-01)
    • Synthesis of Semicyclic Dienes by Modified Julia Olefination of Vinyl Sulfones Derived from Carbohydrates (2007-01-01)
    • Fatty acid profiling and bioactive potential of date palm (Phoenix dactylifera) seed oil: antioxidant, antimicrobial, and α-glucosidase inhibitory activities (2025-01-01)
    • Synthesis, Molecular Docking and Anticancer Activity of New Substituted Pyridine-1,2,3-Triazole Hybrid N-Glycosides Via Click Chemistry (2024-01-01)
    • Optical and photoelectronic properties of a new material: Optoelectronic application (2020-01-01)
    • Unprecedented Synthesis of 4-Ylidene (3S)-3-hydroxy-1-aryl (alkyl)-pyrrolidine-2,5-diones Based on 1,3-Dipolar Cycloaddition of a Sugar-Derived Nitrone to N-Substituted ... (2019-01-01)
    • Evaluation of Antioxidant, Anti-inflammatory, Anti-hemolytic, and Enzyme Inhibitory Activities of Polysaccharide Derived from Opuntia stricta (Haw.) Haw. Pulp and … (2025-01-01)
    • Antioxidant and Antimicrobial Activities of Thyme (Thymus vulgaris L.) Essential Oil Growing Wild in Tunisia (2021-01-01)
    • Anti-ulcer activity of green synthesized selenium nanoparticles using Nigella sativa L. seed extract in rats (2025-01-01)
    • Comprehensive multispectral and computational study of isoxazolidine derivative ‘ISoXD3’: Synthesis, spectral characteristics, DNA binding, and comparative effects of allyl and… (2025-01-01)
    • Synthesis of a novel enantiopure imidazo-isoxazole derivatives and in silico prediction of ADME/pharmacokinetics properties (2023-01-01)
    • Mechanochemical Promoted Heterocycles: A Solvent-Free Route to Triazole Carbohydrates as Glycogen Phosphorylase Inhibitors (2022-01-01)
    • Unprecedented 3-O-methyl-3-C-trifluoromethyl-d-ribono-(and l-lyxono)-γ-lactones synthesized by nucleophilic trifluoromethylation of d-hexose-derived cyclic ketones (2016-01-01)
    • Study of the Regio- and Stereoselectivity of [3+2] Cycloaddition of Nitrile Oxides to Various Racemic 3-acyloxy and 3-hydroxybut-1-enes (2012-01-01)
    • Synthesis of Novel Thiosemicarbazones and Their Molecular Docking Simulations as Inhibitors of α-Amylase and α-Glycosidase Enzymes (2025-01-01)
    • Exploring the antioxidant potency of novel indolin-2-one-based imidazo-isoxazole hybrids: Design, synthesis, and computational studies (2025-01-01)
    • Exploring 1,3-dipolar cycloaddition reactions of nitrones with alkenes: Synthesis of isoxazolidine derivatives (2025-01-01)
    • Design, Characterization, and Molecular Docking Study of New Isoxazolidine-1,2,3-Triazole Hybrids (2024-01-01)
    • S. Ghannay Synthesis of (3S, 3aS, 6aS)-2-acetyl-N-methylhexahydrofuro [3, 4-d][1, 2] oxazole-3-carboxamide via an oxidative cleavage using m-CPBA. ADME approach: Ghannay et al (2022-01-01)
    • Synthesis and characterization of novel isoxazolidine-thiosemicarbazone hybrid derivatives as precursors of unnatural amino acids (2022-01-01)
    • Crystal structure of (1S, 2S, 2′R, 3a′S, 5R)-2′-[(5-bromo-1H-indol-3-yl)methyl]-2-isopropyl-5,5′-dimethyldihydro-2′H-spiro[cyclohexane-1,6′-imidazo[1,5-b… (2016-01-01)
    • Crystal structure of 5-chloromethyl-N-methyl-4-[(4-phenyl-1,2,3-triazol-1-yl)methyl]isoxazolidine-3-carboxamide (2016-01-01)
    • (1S, 2R, 2′ S, 3′a S, 5R)-2′-[(1S)-1-Hydroxyethyl]-2-isopropyl-5, 5′-dimethyl-3′, 3′a-dihydro-2′H-spiro[cyclohexane-1, 6′-imidazo[1, 5-b]isoxazol]-4′(5′H)-one (2007-01-01)
    • Interaction Studies of a Novel Enantiopure Isoxazolidine with DNA and β-Cyclodextrin: Binding and Antioxidant Properties (2026-01-01)
    • Neuroprotective effects of *Artemisia campestris* essential oil against chlorpyrifos-induced toxicity in rats supported by computational modelling (2025-01-01)
    • Protective effect of Arthrocnemum indicum ethanolic extract on hypercholesterolemic rats along with antioxidant and antimicrobial activities (2025-01-01)
    • . Click Chemistry: a promising approach for 1,2,3-triazole synthesis (2024-01-01)
    • Synthesis of New 1,2,3-Triazole Glycoside-Based Quinoline Systems via Click Cycloaddition (2023-01-01)
    • Preparation and characterization of ZnO nanoparticles incorporated by mechanical milling into cellulose for electrical insulator applications (2022-01-01)
    • Synthesis of (3S,3aS,6aS)-2-acetyl-N-methylhexahydrofuro[3,4- d][1,2]oxazole-3-carboxamide via oxidative cleavage using m-CPBA. ADME approach (2022-01-01)
    • Thymus vulgaris L. Essential Oil: Effect on Fatty Acid and Protein Oxidation in Little Tuna (Euthynnus alletteratus) Minced During Refrigerated Storage (2021-01-01)
    • Proceedings of the First Maghrebi Colloquium on Heterocyclic Chemistry: CMCH 1-2017 held on May 16 & 17, 2017 by the Tunisian Association of Heterocyclic Chemistry and its… (2020-01-01)
    • Additional Iconography for the Article: A Stereoselective Method for the Synthesis of Enantiopure 3-Substituted 4-Hydroxyproline Derivatives via 1,3-Dipolar Cycloadditions (2016-01-01)
    • Crystal structure of 2-isopropyl-5,7'-dimethyl-1',3',3a',6',8a',8b'-hexahydrospiro[cyclohexane-1,6'-furo[3,4-d]imidazo[1,5-b]isoxazol]-8'(7'H)-one (2016-01-01)
    • Pyrrolidine derivatives (2015-01-01)
    • Novel pyrrolidine derivatives (2015-01-01)
    • Synthesis of 4-hydroxyisoleucine analogs, a natural hypoglycemic agent (2006-01-01)
    • Synthesis of a novel enantiopure imidazo-isoxazole derivatives and in silico prediction of ADME/pharmacokinetics properties (2023-01-01)
    • Synthesis and SPAR exploration of new semicarbazone-triazole hybrids in search of potent antioxidant, antibacterial, and antifungal agents (2019-02-01)
    • Biological Activities Evaluation of Enantiopure Isoxazolidine Derivatives: In Vitro, In Vivo and In Silico Studies (2019-03-01)
    • Synthesis of New Porphyrin Complexes: Evaluations of Optical, Electrochemical, and Electronic Properties and Application as an Optical Sensor (2019-01-31)
    • SYNTHESIS OF SOME ISOXAZOLIDINE AND ISOXAZOLINE DERIVATIVES USING NITRONE-DERIVED (-)-MENTHONE VIA 1,3-DIPOLAR CYCLOADDITION WITH ALKENES, ALKYNES, AND CYCLOALKENES (2016-11-01)
    • A stereoselective method for the synthesis of enantiopure 3-substituted 4-hydroxyproline derivatives via 1,3-dipolar cycloadditions (2016-08-01)
    • Unexpected synthesis of aziridines under Cu(I)-catalyzed Kinugasa conditions assisted by microwave irradiation (2016-03-01)
    • Novel routes to either racemic or enantiopure α-amino-(4-hydroxy-pyrrolidin-3-yl)acetic acid derivatives and biological evaluation of a new promising pharmacological scaffold (2015-06-15)
    • Stereoselective Synthesis of Enantiopure Cycloalkylglycines via 1,3-Dipolar Cycloaddition of a Chiral Nitrone to Cycloalkenes (2014-09-01)
    • A Cycloaddition-Cyclization Combined Approach to Enantiopure 3-Glycinyl-4-hydroxypyrrolidines and 3-Substituted 4-Hydroxyprolines (2014-07-01)
    • Stereoselective synthesis of 1,2,3-triazolyl-functionalized isoxazolidines via two consecutive 1,3-dipolar cycloadditions as precursors of unnatural amino acids (2013-04-10)
    • 1,3-Dipolar cycloaddition of a chiral nitrone to (E)-1,4-dichloro-2-butene: a new, efficient synthesis of (2S,3S,4R)-4-hydroxyisoleucine (2012-06-06)
    • Cycloaddition of a chiral nitrone to allylic motifs: a route to enantiopure sugar-based amino acids with a stable glycosidic bond and to 4(S)-4-hydroxy-L-ornithine (2012-02-11)
    • Study of the Regio- and Stereoselectivity of [3+2] Cycloaddition of Nitrile Oxides to Various Racemic 3-acyloxy- and 3-hydroxybut-1-enes (2012-02-01)
    • Inhibition of HSP90 with Pochoximes: SAR and Structure-Based Insights (2009-11-23)
    • Multi-Step Synthesis and Biological Evaluation of Analogs of the Insulin Secretagogue (2S,3R,4S)-4-Hydroxyisoleucine (2009-01-01)
    • Analogs of the insulin secretagogue (2S,3R,4S)-4-hydroxyisoleucine: Synthesis by 1,3-dipolar cycloaddition reactions of chiral nitrones to alkenes (2008-05-16)
    • Divergent synthesis of a pochonin library targeting HSP90 and in vivo efficacy of an identified inhibitor (2008-01-01)
    • C-Glycosyl-Amino-Substituted Hydro- and Benzoquinones: Synthesis and Preliminary Biological Evaluation (2007-11-16)
    • New Synthetic Routes for the Preparation of Enantiopure (2S,3R,4R)-4-Hydroxyisoleucine via 1,3-Dipolar Cycloaddition of a Chiral Nitrone to C4 Alkenes (2007-11-02)
    • Synthesis of semicyclic dienes by modified Julia olefination of vinyl sulfones derived from carbohydrates (2007-10-01)
    • (1S, 2R, 2′S, 3′aS, 5R)-2′-[(1R)-1-hydroxyethyl]-2-isopropyl-5,5′-dimethyl-3′,3′a-dihydro-2′H-spiro[cyclohexane-1,6′-imidazo[1,5-b]isoxazol]4′(5′H)-one (2007-03-01)
    • (1S, 2R, 2′S, 3′aS, 5R)-2′-[(1S)-1-hydroxyethyl]-2-isopropyl-5,5′-dimethyl-3′,3′a-dihydro-2′H-spiro[cyclohexane-1,6′-imidazo[1,5-b]isoxazol]-4′(5′H)-one (2007-03-01)
    • Cycloadditions of chiral nitrones to racemic 3-substituted butenes: Direct access with kinetic resolution to enantiopure dihydroxylated amino acids (2006-12-01)
    • Design, synthesis, biological evaluation, kinetic studies, and molecular modeling of imidazo-isoxazole derivatives targeting both α-amylase and α-glucosidase inhibitors (2024-10-12)
    • Synthesis, optical properties, DNA, β-cyclodextrin interaction, hydrogen isotope sensor, and computational study of a new enantiopure isoxazolidine derivative (ISoXD) (2024-02-17)
    • Identification of dual-target isoxazolidine-isatin hybrids with antidiabetic potential: Design, synthesis, in vitro, and multiscale molecular modeling approaches (2024-02-13)
    • In Silico Design, Synthesis, and Evaluation of Novel Enantiopure Isoxazolidines as Promising Dual Inhibitors of α-Amylase and α-Glucosidase (2024-01-01)
    • In Vitro and In Silico Evaluation of Antiproliferative Activity of New Isoxazolidine Derivatives Targeting EGFR: Design, Synthesis, Cell Cycle Analysis, and Apoptotic Inducers (2023-07-01)
    • Synthesis, optical properties, DNA, β-cyclodextrin interactions, and antioxidant evaluation of a novel isoxazolidine derivative (ISoXD2): A multispectral and computational analysis (2024-07-16)
    • A Reversible Optical Sensor Film for Mercury Ion Discrimination Based on an Isoxazolidine Derivative and Exhibiting pH Sensing (2022-11-01)
    • Design, synthesis, biological evaluation and in silico studies of novel 1,2,3-triazole linked benzoxazine-2,4-dione conjugates as potent antimicrobial, antioxidant and anti-inflammatory agents (vol 15, 104226, 2022) (2023-06-15)
    • Design, synthesis, biological evaluation, and in silico studies of novel 1,2,3-triazole-linked benzoxazine-2,4-dione conjugates as potent antimicrobial, antioxidant, and anti-inflammatory agents (2022-09-11)
    • Multifunctional isoxazolidine derivatives as α-amylase and α-glucosidase inhibitors (2020-05-01)
    • Unprecedented Synthesis of 4-Ylidene (3S)-3-hydroxy-1-aryl(alkyl)-pyrrolidine-2,5-diones via 1,3-Dipolar Cycloaddition of a Sugar-Derived Nitrone to N-Substituted Maleimides (2019-05-24)
    • GC/MS Profiling, Antibacterial, Anti-Quorum Sensing, and Antibiofilm Properties of Anethum graveolens L. Essential Oil: A Molecular Docking Study and In Silico ADME Profiling (2023-05-16)
    • Multifunctional Derivatives of Spiropyrrolidine Tethered Indeno-Quinoxaline Heterocyclic Hybrids as Potent Antimicrobial, Antioxidant, and Antidiabetic Agents: Design, Synthesis, In Vitro, and In Silico Approaches (2022-11-01)
    • In Vitro and In Silico Screening of the Anti-Vibrio spp., Antibiofilm, Antioxidant, and Anti-Quorum Sensing Activities of Cuminum cyminum L. Volatile Oil (2022-09-01)
    • Phytochemical Profiling, Antimicrobial and α-Glucosidase Inhibitory Potential of Phenolic-Enriched Extracts from the Aerial Parts of Echium humile Desf.: An In Vitro Study Combined with an In Silico Approach (2022-05-01)
    • GC-MS Profiling, Vibriocidal, Antioxidant, Antibiofilm, and Anti-Quorum Sensing Properties of Carum carvi L. Essential Oil: In Vitro and In Silico Approaches (2022-04-01)
    • Phytochemical Profiling of the Aqueous Extract of Allium subhirsutum L. with Antioxidant, Antimicrobial, Antibiofilm, and Anti-Quorum Sensing Properties: In Vitro and In Silico Studies (2022-02-01)
    • HPLC-MS Profiling and Antioxidant, Antimicrobial, Antidiabetic, and Cytotoxic Activities of Arthrocnemum indicum (Willd.) Moq. Extracts (2022-01-01)
    • HPLC/MS Phytochemical Profiling and Antioxidant Activities of Echium humile Desf. Extracts: ADMET Prediction and a Computational Study Targeting the Human Peroxiredoxin 5 Receptor (2021-11-01)
    • Novel enantiopure isoxazolidine and C-alkyl imine oxide derivatives as potential hypoglycemic agents: Design, synthesis, dual inhibitors of α-amylase and α-glucosidase, ADMET, and molecular docking study (2020-11-01)
    • Design, Synthesis, Molecular Properties, and In Vitro Antioxidant and Antibacterial Potential of Novel Enantiopure Isoxazolidine Derivatives (2020-01-01)
    • Stereoselective Synthesis of Enantiopure N-Substituted Pyrrolidin-2,5-dione Derivatives via 1,3-Dipolar Cycloaddition and Evaluation of Their In Vitro Antioxidant and Antibacterial Activities (2017-06-01)
    • Unprecedented stereoselective synthesis of 3-methylisoxazolidine-5-aryl-1,2,4-oxadiazoles via 1,3-dipolar cycloaddition and study of their in vitro antioxidant activity (2016-01-01)
    • Unprecedented 3-O-methyl-3-C-trifluoromethyl-D-ribono- (and L-lyxono)-γ-lactones synthesized by nucleophilic trifluoromethylation of D-hexose-derived cyclic ketones (2016-06-01)
    • Advanced Synthetic Strategies and Therapeutic Applications of Nitrogen Heterocyclic Compounds (2026-01-01)
    • Synthesis, Photophysical and Docking Studies of a Novel Isoxazolidine–Benzimidazole Hybrid and Preliminary Cytotoxic Evaluation: Binding Interactions with DNA and β-Cyclodextrin (2026-01-01)
    • From Surface Engineering to Targeted Nanomedicine: The Evolving Role of Gold Nanoparticles (2026-01-01)
    • Synthesis, photophysical and docking studies of a novel isoxazolidine-benzimidazole hybrid and preliminary cytotoxic evaluation: Binding interactions with DNA and β-cyclodextrin (2026-12-15)
    • Exploring the antioxidant potency of novel indolin-2-one-based imidazo-isoxazole hybrids: Design, synthesis, and computational studies (2026-02-05)
    • Neuroprotective effects of *Artemisia campestris* essential oil against chlorpyrifos-induced toxicity in rats supported by computational modelling (2026-01-01)
    • Evaluation of Antioxidant, Anti-inflammatory, Anti-hemolytic, and Enzyme Inhibitory Activities of Polysaccharide Derived from Opuntia stricta (Haw.) Pulp and its Effects on Wound Healing in Diabetic Rats (2025-12-01)
    • Untargeted metabolomics approach based on UPLC-ESI-QTOF-MS/MS and evaluation of antioxidant and cytotoxic activities of Nepeta deflersiana Schweinf. ex Hedge supported by molecular modeling and ADMET analysis (2025-06-25)
    • Protective effect of Arthrocnemum indicum ethanolic extract on hypercholesterolemic rats along with antioxidant and antimicrobial activities (2025-06-01)
    • Fatty acid profiling and bioactive potential of date palm (Phoenix dactylifera) seed oil: antioxidant, antimicrobial, and α-glucosidase inhibitory activities (2025-04-01)
    • Comprehensive multispectral and computational study of isoxazolidine derivative ‘ISoXD3’: Synthesis, spectral characteristics, DNA binding, and comparative effects of allyl and propargyl groups on optical properties (2025-03-01)
    • Anti-ulcer activity of green synthesized selenium nanoparticles using Nigella sativa L. seed extract in rats (2025-01-01)
    • GC-MS/MS Analysis and Wound Repair Potential of Urtica dioica Essential Oil: In silico Modeling and In vivo Study in Rats (2025-01-01)
    • Synthesis, Molecular Docking, and Anticancer Activity of New Substituted Pyridine-1,2,3-Triazole Hybrid N-Glycosides via Click Chemistry (2024-12-01)
    • Design, synthesis, biological evaluation, kinetic studies, and molecular modeling of imidazo-isoxazole derivatives targeting both α-amylase and α-glucosidase inhibitors (2024-10-30)
    • Synthesis, optical properties, DNA, β-cyclodextrin interactions, and antioxidant evaluation of a novel isoxazolidine derivative (ISoXD2): A multispectral and computational analysis (2024-07-30)
    • Synthesis, photophysical and docking studies of a novel isoxazolidine–benzimidazole hybrid and preliminary cytotoxic evaluation: Binding interactions with DNA and β-cyclodextrin (2026-12-15)
    • Identification of dual-target isoxazolidine-isatin hybrids with antidiabetic potential: Design, synthesis, in vitro, and multiscale molecular modeling approaches (2024-02-29)
    • Synthesis, optical properties, DNA, β-cyclodextrin interaction, hydrogen isotope sensor, and computational study of a new enantiopure isoxazolidine derivative (ISoXD) (2024-02-29)
    • In Silico Design, Synthesis, and Evaluation of Novel Enantiopure Isoxazolidines as Promising Dual Inhibitors of α-Amylase and α-Glucosidase (2024-01-01)
    • Corrigendum to “Design, synthesis, biological evaluation and in silico studies of novel 1,2,3-triazole-linked benzoxazine-2,4-dione conjugates as potent antimicrobial, antioxidant and anti-inflammatory agents” [Arab. J. Chem. 15(11) (2022) 104226](S1878535222005421)(10.1016/j.arabjc.2022.104226) (2023-09-01)
    • In Vitro and In Silico Evaluation of Antiproliferative Activity of New Isoxazolidine Derivatives Targeting EGFR: Design, Synthesis, Cell Cycle Analysis, and Apoptotic Inducers (2023-07-01)
    • GC/MS Profiling, Antibacterial, Anti-Quorum Sensing, and Antibiofilm Properties of Anethum graveolens L. Essential Oil: Molecular Docking Study and In-Silico ADME Profiling (2023-05-01)
    • Phytochemical profiling, antimicrobial, antibiofilm, insecticidal, and anti-leishmanial properties of aqueous extract from Juglans regia L. root bark: In vitro and in silico approaches (2023-01-01)
    • Synthesis of a novel enantiopure imidazo-isoxazole derivatives and in silico prediction of ADME/pharmacokinetics properties (2023-01-01)
    • Mechanochemical promoted heterocycles: A solvent-free route to triazole carbohydrates as glycogen phosphorylase inhibitors (2022-12-01)
    • A Reversible Optical Sensor Film for Mercury Ion Discrimination Based on an Isoxazolidine Derivative and Exhibiting pH Sensing (2022-11-01)
    • Multifunctional Derivatives of Spiropyrrolidine Tethered Indeno-Quinoxaline Heterocyclic Hybrids as Potent Antimicrobial, Antioxidant, and Antidiabetic Agents: Design, Synthesis, In Vitro, and In Silico Approaches (2022-11-01)
    • Design, synthesis, biological evaluation and in silico studies of novel 1,2,3-triazole-linked benzoxazine-2,4-dione conjugates as potent antimicrobial, antioxidant and anti-inflammatory agents (2022-11-01)
    • Design, synthesis, in vitro anticancer and antimicrobial evaluation, SAR analysis, molecular docking and dynamic simulation of new pyrazoles, triazoles and pyridazines based isoxazole (2022-09-15)
    • Novel (2-Oxoindolin-3-ylidene)methyl)-1H-pyrazole and their fused derivatives: Design, synthesis, antimicrobial evaluation, DFT, chemical approach, in silico ADME and molecular docking studies (2022-09-15)
    • In Vitro and In Silico Screening of Anti-Vibrio spp., Antibiofilm, Antioxidant and Anti-Quorum Sensing Activities of Cuminum cyminum L. Volatile Oil (2022-09-01)
    • Synthesis and Characterization of Novel Isoxazolidine-Thiosemicarbazone Hybrid Derivatives as Precursor of Unnatural Amino Acids (2022-09-01)
    • Phytochemical Profiling, Antimicrobial and α-Glucosidase Inhibitory Potential of Phenolic-Enriched Extracts of the Aerial Parts from Echium humile Desf.: In Vitro Combined with In Silico Approach (2022-05-01)
    • New Spiropyrrolothiazole Derivatives Bearing an Oxazolone Moiety as Potential Antidiabetic Agents: Design, Synthesis, Crystal Structure, Hirshfeld Surface Analysis, ADME, and Molecular Docking Studies (2022-04-15)
    • Preparation and characterization of ZnO nanoparticles incorporated by mechanical milling into cellulose for electrical insulator applications (2022-04-01)
    • GC-MS Profiling, Vibriocidal, Antioxidant, Antibiofilm, and Anti-Quorum Sensing Properties of Carum carvi L. Essential Oil: In Vitro and In Silico Approaches (2022-04-01)
    • Phytochemical Profiling of Allium subhirsutum L. Aqueous Extract with Antioxidant, Antimicrobial, Antibiofilm, and Anti-Quorum Sensing Properties: In Vitro and In Silico Studies (2022-02-01)
    • HPLC-MS Profiling, Antioxidant, Antimicrobial, Antidiabetic, and Cytotoxicity Activities of Arthrocnemum indicum (Willd.) Moq. Extracts (2022-01-01)
    • Emetine, a potent alkaloid for the treatment of SARS-CoV-2 targeting papain-like protease and non-structural proteins: pharmacokinetics, molecular docking and dynamic studies (2022-01-01)
    • Towards a treatment of antibacterial and antifungal infections: Design, synthesis and in vitro activity of novel arylhydrazothiazolylsulfonamide analogues and their insight of DFT, docking and molecular dynamic simulations (2021-11-05)
    • Hplc/ms phytochemical profiling with antioxidant activities of echium humile desf. Extracts: Admet prediction and computational study targeting human peroxiredoxin 5 receptor (2021-11-01)
    • X-ray molecular structure characterization of a hexamethylenetetramine zinc(II) porphyrin complex, catalytic degradation of toluidine blue dye, experimental and statistical studies of adsorption isotherms (2021-11-01)
    • Tomatidine and patchouli alcohol as inhibitors of SARS-CoV-2 enzymes (3CLpro, PLpro, and NSP15) by molecular docking and molecular dynamics simulations (2021-10-01)
    • Synthesis, Structure-Activity Relationship and in silico Studies of Novel Pyrazolothiazole and Thiazolopyridine Derivatives as Prospective Antimicrobial and Anticancer Agents (2021-08-20)
    • Antimicrobial, antioxidant, anti-acetylcholinesterase, antidiabetic, and pharmacokinetic properties of carum carvi l. And coriandrum sativum l. essential oils alone and in combination (2021-06-02)
    • Bioactivities and in silico study of Pergularia tomentosa L. phytochemicals as potent antimicrobial agents targeting type IIA topoisomerase, TyrRS, and Sap1 virulence proteins (2021-05-01)
    • LC-ESI/MS-Phytochemical profiling with antioxidant, antibacterial, antifungal, antiviral and in silico pharmacological properties of Algerian asphodelus tenuifolius (Cav.) organic extracts (2021-04-01)
    • New substituted pyrazolones and dipyrazolotriazines as promising tyrosyl-tRNA synthetase and peroxiredoxin-5 inhibitors: Design, synthesis, molecular docking, and structure-activity relationship (SAR) analysis (2021-04-01)
    • Repurposing of anisomycin and oleandomycin as potential anti-SARS-CoV-2 virus agents targeting key enzymes using virtual computational approaches (2021-01-01)
    • Tripeptides from Allium subhirsutum L. extracts: Pharmacokinetic properties, toxicity prediction, and in silico study against SARS-CoV-2 enzymes and pro-inflammatory proteins (2021-01-01)
    • Novel fused pyridine derivatives containing a pyrimidine moiety as prospective tyrosyl-tRNA synthetase inhibitors: Design, synthesis, pharmacokinetics, and molecular docking studies (2020-11-05)
    • Antioxidant activities of a new chemotype of piper cubeba L. Fruit essential oil (methyleugenol/eugenol): In silico molecular docking and admet studies (2020-11-01)
    • Hr-lcms-based metabolite profiling, antioxidant, and anticancer properties of teucrium polium l. Methanolic extract: Computational and in vitro study (2020-11-01)
    • Novel enantiopure isoxazolidine and C-alkyl imine oxide derivatives as potential hypoglycemic agents: Design, synthesis, dual inhibitors of α-amylase and α-glucosidase, ADMET and molecular docking study (2020-11-01)
    • Allium subhirsutum L. As a potential source of antioxidant and anticancer bioactive molecules: Hr-lcms phytochemical profiling, in vitro and in vivo pharmacological study (2020-10-01)
    • Design, synthesis, ADMET, and molecular docking of new imidazo[4,5-b]pyridine-5-thione derivatives as potential tyrosyl-tRNA synthetase inhibitors (2020-09-01)
    • Zinc(ii) triazole: Meso-arylsubstituted porphyrins for UV-visible chloride and bromide detection. Adsorption and catalytic degradation of malachite green dye (2020-06-12)
    • In vitro antimicrobial and α-glucosidase inhibitory potential of enantiopure cycloalkylglycine derivatives: Insights into their in silico pharmacokinetic, druglikeness, and medicinal chemistry properties (2020-06-01)
    • Multifunctional isoxazolidine derivatives as α-amylase and α-glucosidase inhibitors (2020-05-01)
    • Effect of the coordination of π-acceptor 4-cyanopyridine ligand on the structural and electronic properties of: Meso-tetra(para-methoxy) and meso-tetra(para-chlorophenyl) porphyrin cobalt(ii) coordination compounds. Application in the catalytic degradation of methylene blue dye (2020-02-01)
    • Synthesis, in vitro antimicrobial assessment, and computational investigation of pharmacokinetic and bioactivity properties of novel trifluoromethylated compounds using in silico ADME and toxicity prediction tools (2020-02-01)
    • Optical and photoelectronic properties of a new material: Optoelectronic application (2020-01-01)
    • Unprecedented Synthesis of 4-Ylidene (3 S)-3-hydroxy-1-aryl (alkyl)-pyrrolidine-2,5-diones Based on 1,3-Dipolar Cycloaddition of a Sugar-derived Nitrone to N-Substituted Maleimides (2019-05-24)
    • Synthesis and SPAR exploration of new semicarbazone-triazole hybrids in search of potent antioxidant, antibacterial, and antifungal agents (2019-02-01)
    • Synthesis of New Porphyrin Complexes: Evaluations of Optical, Electrochemical, and Electronic Properties and Application as an Optical Sensor (2019-01-31)
    • Design, synthesis, molecular properties, and in vitro antioxidant and antibacterial potential of novel enantiopure isoxazolidine derivatives (2020-01-01)
    • Biological Activities Evaluation of Enantiopure Isoxazolidine Derivatives: In Vitro, In Vivo and In Silico Studies (2019-03-15)
    • Stereoselective synthesis of enantiopure N-substituted pyrrolidin-2,5-dione derivatives by 1,3-dipolar cycloaddition and assessment of their in vitro antioxidant and antibacterial activities (2017-01-01)
    • Crystal structure of (1S,2S,2'R,3a'S,5R)-2'-[(5-bromo-1H-indol-3-yl)methyl]-2-isopropyl-5,5'-dimethyldihydro-2'H-spiro[cyclohexane-1,6'-imidazo[1,5-b]isoxazole]-4'(5'H)-one (2016-08-01)
    • Crystal structure of 2-isopropyl-5,7'-dimethyl-1',3',3a',6',8a',8b'-hexahydrospiro[cyclohexane-1,6'-furo[3,4-d]imidazo[1,5-b]isoxazol]-8'(7'H)-one (2016-08-01)
    • A stereoselective method for the synthesis of enantiopure 3-substituted 4-hydroxyproline derivatives via 1,3-dipolar cycloadditions (2016-08-01)
    • Unprecedented 3-O-methyl-3-C-trifluoromethyl-d-ribono- (and l-lyxono)-γ-lactones synthesized by nucleophilic trifluoromethylation of d-hexose-derived cyclic ketones (2016-06-01)
    • Unexpected synthesis of aziridines under Cu(I)-catalyzed Kinugasa conditions assisted by microwave irradiation (2016-03-01)
    • Unprecedented stereoselective synthesis of 3-methylisoxazolidine-5-aryl-1,2,4-oxadiazoles via 1,3-dipolar cycloaddition and study of their in vitro antioxidant activity (2016-01-01)
    • Synthesis of some isoxazolidine and isoxazoline derivatives using nitrone-derived (-)-menthone via 1,3-dipolar cycloaddition with alkenes, alkynes and cycloalkenes (2016-01-01)
    • Crystal structure of 5-chloromethyl-N-methyl-4-[(4-phenyl-1,2,3-triazol-1-yl)methyl]isoxazolidine-3-carboxamide (2016-01-01)
    • Novel routes to either racemic or enantiopure α-amino-(4-hydroxy-pyrrolidin-3-yl)acetic acid derivatives and biological evaluation of a new promising pharmacological scaffold (2015-05-31)
    • Stereoselective synthesis of enantiopure cycloalkylglycines by 1,3-dipolar cycloaddition of a chiral nitrone to cycloalkenes (2014-01-01)
    • A cycloaddition-cyclization combined approach to enantiopure 3-glycinyl-4-hydroxypyrrolidines and 3-substituted 4-hydroxyprolines (2014-01-01)
    • Stereoselective synthesis of 1,2,3-triazolyl-functionalized isoxazolidines via two consecutive 1,3-dipolar cycloadditions as precursors of unnatural amino acids (2013-04-10)
    • 1,3-Dipolar cycloaddition of a chiral nitrone to (E)-1,4-dichloro-2-butene: A new efficient synthesis of (2S,3S,4R)-4-hydroxyisoleucine (2012-06-06)
    • Cycloaddition of a chiral nitrone to allylic motifs: An access to enantiopure sugar-based amino acids displaying a stable glycosidic bond and to 4(S)-4-hydroxy-l-ornithine (2012-02-11)
    • Study of the regio- and stereoselectivity of [3+2] cycloaddition of nitrile oxides to various racemic 3-acyloxy and 3-hydroxybut-1-enes (2012-02-01)
    • Inhibition of HSP90 by pochoximes: SAR and structure-based insights (2009-11-23)
    • Multi-step synthesis and biological evaluation of analogues of insulin secretagogue (2S,3R,4S)-4-hydroxyisoleucine (2009-01-01)
    • Divergent synthesis of a pochonin library targeting HSP90 and in vivo efficacy of an identified inhibitor (2008-05-26)
    • Analogues of insulin secretagogue (2S,3R,4S)-4-hydroxyisoleucine: synthesis by 1,3-dipolar cycloaddition reactions of chiral nitrones to alkenes (2008-05-16)
    • C-glycosyl amino-substituted hydro- and benzoquinones: Synthesis and preliminary biological evaluation (2007-11-16)
    • New synthetic routes toward enantiopure (2S,3R,4R)-4-hydroxyisoleucine by 1,3-dipolar cycloaddition of a chiral nitrone to C4 alkenes (2007-11-02)
    • Synthesis of semicyclic dienes by modified Julia olefination of vinyl sulfones derived from carbohydrates (2007-10-01)
    • (1S,2R,2′S,3′aS,5R)-2′-[(1S)-1-hydroxyethyl] -2-isopropyl-5,5′-dimethyl-3′,3′a-dihydro-2′H-spiro-[cyclohexane-1,6′-imidazo[1,5-b]isoxazole]-4′(5′H)-one (2007-02-28)
    • (1S,2R,2′S,3′aS,5R)-2′-[(1R)-1-hydroxyethyl] -2-isopropyl-5,5′-dimethyl-3′,3′a-dihydro-2′H-spiro-[cyclohexane-1,6′-imidazo[1,5-b]isoxazole]-4′(5′H)-one (2007-02-28)
    • Cycloadditions of chiral nitrones to racemic 3-substituted butenes: Direct access with kinetic resolution to enantiopure dihydroxylated amino acids (2006-12-01)
    • Ginger essential oil as a green nanotechnology agent: Composition, nanoparticle synthesis, and biomedical applications (2025-01-01)

    Teaching materials

    • General Chemistry Chem 202
    • Advanced Organic Chemistry Chem 640
    • Kim Spectra 442
    • Organic Chemistry Chem 249
    • Organic Chemistry 2. Chem340

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